E7016

Product Name: E7016
Description: E7016, also known as GPI21016, is an inhibitor of the nuclear enzyme poly (ADP-ribose) polymerase (PARP) with potential chemo- and/or radiosensitizing activity. PARP inhibitor E7016 selectively binds to PARP and prevents PARP-mediated DNA repair of singl
CAS NO: 329689-23-8 Product: Monastrol
Synonym: E7016; E-7016; E 7016; GPI21016; GPI 21016; GPI-21016.
IUPAC Chemical Name: 10-((4-Hydroxypiperidin-1-yl)methyl)chromeno[4,3,2-de]phthalazin-3(2H)-one
In ChiKey: HAVFFEMDLROBGI-UHFFFAOYSA-NVEGFR inhibitors
SMILE Code: O=C1NN=C2C3=C1C=CC=C3OC4=C2C=C(CN5CCC(O)CC5)C=C4
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 5 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22118433
Chemical Formula:C20H19N3O3
ExactMass: 349.14264
Molecular Weight: 349.383
Elemental Analysis: C, 68.75; H, 5.48; N, 12.03; O, 13.74

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