Product Name: P505-15 hydrochloride featured
Description: P505-15, also known as PRT2607, PRT062607, and BIIB057, is a novel, highly selective, and orally bioavailable small molecule SYK inhibitor (SYK IC(50) = 1 nM) with anti-SYK activity that is at least 80-fold greater than its affinity for other kinases. P50
CAS NO: 1239875-86-5 Product: SGI-7079
Synonym: PRT2607; PRT-2607; PRT 2607; PRT062607; PRT-062607; PRT 062607; P-505-15; P 505-15; P505-15; BIIB057; BIIB-057; BIIB 057.
IUPAC Chemical Name: 4-((3-(2H-1,2,3-triazol-2-yl)phenyl)amino)-2-(((1R,2S)-2-aminocyclohexyl)amino)pyrimidine-5-carboxamide hydrochloride
In ChiKey: RMNLLPXCNDZJMJ-IDVLALEDSA-NSigma Receptor inhibitors
SMILE Code: O=C(C1=CN=C(N[C@H]2[C@@H](N)CCCC2)N=C1NC3=CC=CC(N4N=CC=N4)=C3)N.[H]Cl
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22138732
Chemical Formulaļ¼C19H24ClN9O
ExactMass: 393.20256
Molecular Weight: 429.913
Elemental Analysis: C, 53.08; H, 5.63; Cl, 8.25; N, 29.32; O, 3.72
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