A-395

Product Name: A-395
Description: A-395 is a potent and selective EED inhibitor. A-395 includes potent binding to EED with Ki = 0.4 nM, inhibits the PRC2 complex with IC50 = 34 nM for methylation of H3K27 and greater than 100-fold selectivity over other histone methyltransferases and non
CAS NO: 106612-94-6 Product: GLP-1(7-37)
Synonym: A-395; A 395; A395.
IUPAC Chemical Name: (3R,4S)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)-N,N-dimethyl-4-(4-(4-(methylsulfonyl)piperazin-1-yl)phenyl)pyrrolidin-3-amine
In ChiKey: REVJNSVNICWODC-KIDMSAQOSA-NAdenosine Receptor inhibitors
SMILE Code: CN([[email protected]]1CN(C2CCC3=C2C(F)=CC=C3)C[C@@H]1C4=CC=C(N5CCN(S(=O)(C)=O)CC5)C=C4)C
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22110401
Chemical Formula:C26H35FN4O2S
ExactMass: 486.2465
Molecular Weight: 486.6504
Elemental Analysis: C, 64.17; H, 7.25; F, 3.90; N, 11.51; O, 6.58; S, 6.59

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A-395

Product Name: A-395
Description: A-395 is a potent and selective EED inhibitor. A-395 includes potent binding to EED with Ki = 0.4 nM, inhibits the PRC2 complex with IC50 = 34 nM for methylation of H3K27 and greater than 100-fold selectivity over other histone methyltransferases and non
CAS NO: 106612-94-6 Product: GLP-1(7-37)
Synonym: A-395; A 395; A395.
IUPAC Chemical Name: (3R,4S)-1-(7-fluoro-2,3-dihydro-1H-inden-1-yl)-N,N-dimethyl-4-(4-(4-(methylsulfonyl)piperazin-1-yl)phenyl)pyrrolidin-3-amine
In ChiKey: REVJNSVNICWODC-KIDMSAQOSA-NAdenosine Receptor inhibitors
SMILE Code: CN([[email protected]]1CN(C2CCC3=C2C(F)=CC=C3)C[C@@H]1C4=CC=C(N5CCN(S(=O)(C)=O)CC5)C=C4)C
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22110401
Chemical Formula:C26H35FN4O2S
ExactMass: 486.2465
Molecular Weight: 486.6504
Elemental Analysis: C, 64.17; H, 7.25; F, 3.90; N, 11.51; O, 6.58; S, 6.59

About author

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You must be logged in to post a comment.