Fasitibant chloride (HCl salt)

Product Name: Fasitibant chloride (HCl salt)
Description: Fasitibant chloride, also known as MEN16132, is a potent and selective nonpeptide kinin B2 receptor antagonist. MEN16132 inhibited in a dose-dependent manner the bronchoconstriction induced by BK (10 nmol/kg i.v.). MEN16132 was more potent and possessed a
CAS NO: 701977-08-4 Product: Taranabant ((1R,2R)stereoisomer)
Synonym: MEN16132; MEN-16132; MEN 16132; Fasitibant chloride
IUPAC Chemical Name: (S)-4-amino-5-(4-(4-((2,4-dichloro-3-(((2,4-dimethylquinolin-8-yl)oxy)methyl)phenyl)sulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-5-oxopentan-1-aminium chloride hydrochloride
In ChiKey: Steroids inhibitors
SMILE Code: O=C(N1CCN(C(C2(NS(=O)(C3=CC=C(Cl)C(COC4=C5N=C(C)C=C(C)C5=CC=C4)=C3Cl)=O)CCOCC2)=O)CC1)[C@@H](N)CCC[N+](C)(C)C.[H]Cl.[Cl-]
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22120389
Chemical Formulaļ¼šC36H50Cl4N6O6S
ExactMass:
Molecular Weight: 836.692
Elemental Analysis: C, 51.68; H, 6.02; Cl, 16.95; N, 10.04; O, 11.47; S, 3.83

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