Product Name: Dapitant
Description: Dapitant, also known as RPR100893, is potent and selective NK1 receptor antagonist both in vitro and in vivo, and exhibits high affinity for guinea pig and human NK1 receptor . Dapitant was developed as a potential drug for the acute treatment of migraine
CAS NO: 1627696-51-8 Product: LY3177833
Synonym: RPR100893; RPR 100893; RPR-100893; Erispant; Dapitant.
IUPAC Chemical Name: (S)-1-((3aS,4S,7aS)-4-hydroxy-4-(2-methoxyphenyl)-7,7-diphenylhexahydro-1H-isoindol-2(3H)-yl)-2-(2-methoxyphenyl)propan-1-one
In ChiKey: PIKfyve inhibitors
SMILE Code: C[[email protected]@H](C1=CC=CC=C1OC)C(N2C[[email protected]]3([H])C(C4=CC=CC=C4)(C5=CC=CC=C5)CC[[email protected]](C6=CC=CC=C6OC)(O)[[email protected]]3([H])C2)=O
Appearance: white solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/2211736
Chemical Formulaļ¼šC37H39NO4
ExactMass: 561.28791
Molecular Weight: 561.70986
Elemental Analysis: C, 79.11; H, 7.00; N, 2.49; O, 11.39