Product Name: Obicetrapib (free base)
Description: Obicetrapib (also known as AMG-899, TA-8995, and DEX-001) is a cholesteryl ester transfer protein (CETP) inhibitor. CETP inhibitors substantially increase the concentration of high-density lipoprotein cholesterol (HDL-C), which may have a possible benefic
CAS NO: 10083-24-6 Product: Piceatannol
Synonym: Obicetrapib; AMG-899, TA-8995, DEZ-001; AMG 899, TA 8995, DEZ 001; AMG899, TA8995, DEZ001; 866399-87-3 (free base); 866399-89-5 (calcium)
IUPAC Chemical Name: 4-((2-((3,5-bis(trifluoromethyl)benzyl)((2R,4S)-1-(ethoxycarbonyl)-2-ethyl-6-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)pyrimidin-5-yl)oxy)butanoic acid
In ChiKey: 5-HT Receptor inhibitors
SMILE Code: O=C(O)CCCOC1=CN=C(N(CC2=CC(C(F)(F)F)=CC(C(F)(F)F)=C2)[C@H]3C[C@@H](CC)N(C(OCC)=O)C4=C3C=C(C(F)(F)F)C=C4)N=C1
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22137330
Chemical Formulaļ¼C32H31F9N4O5
ExactMass: 722.2151
Molecular Weight: 722.6086
Elemental Analysis: C, 53.19; H, 4.32; F, 23.66; N, 7.75; O, 11.07
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